SCHEMBL26550554

SCHEMBL26550554

CC(C)Nc1cc(N2CCOCC2)ccn1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.59
CHEK1 O14757 10/20 0.53
NPY1R P25929 1/20 0.46
KCNH2 Q12809 1/20 0.46
LRRK2 Q5S007 2/20 0.45
CSF1R P07333 1/20 0.45
PDGFRA P16234 1/20 0.45
ATR Q13535 1/20 0.44
ATRIP Q8WXE1 1/20 0.44
MAPK10 P53779 1/20 0.43
CDK4 P11802 1/20 0.43
CCNA2 P20248 1/20 0.43
CCND1 P24385 1/20 0.43
CDK2 P24941 1/20 0.43
CCND3 P30281 1/20 0.43
CDK6 Q00534 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25493009 0.84 HRH4 (0.68) HRH4LRRK2
SCHEMBL25769210 0.83 CHEK1 (0.53) HRH4CHEK1MAPK10
SCHEMBL25493007 0.82 HRH4 (0.69) HRH4CHEK1
SCHEMBL19699523 0.80 MTOR (0.49) CHEK1MAPK10
Hydrochloric Acid SCHEMBL4721451 0.79 CHEK1 (0.49) HRH4CHEK1MAPK10CDK2
SCHEMBL26572368 0.78 PCSK9 (0.54) LRRK2CSF1RPDGFRACDK4CCNA2
SCHEMBL19706560 0.77 ADORA2A (0.59) CHEK1KCNH2MAPK10
SCHEMBL807537 0.77 CHEK1 (0.47) CHEK1LRRK2CDK2
SCHEMBL25292457 0.75 MTOR (0.53) CHEK1MAPK10
SCHEMBL847015 0.75 HRH4 (0.72) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023196975-A1 COMPOUNDS THAT INTERACT WITH RAS SUPERFAMILY PROTEINS FOR TREATMENT OF CANCERS, INFLAMMATORY DISEASES, RASOPATHIES, AND FIBROTIC DISEASE SHY THERAPEUTICS, LLC (US) 2023-10-12 WO disclosed