SCHEMBL2655813

SCHEMBL2655813

CC(COc1ccc(Cl)cn1)C(=O)NC(C)C(Cc1ccc(Cl)cc1)c1ccsc1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 18/20 0.52
CNR2 P34972 11/20 0.52
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
KCNH2 Q12809 1/20 0.40
FDFT1 P37268 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1900604 0.83 CNR1 (0.77) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL2246652 0.75 CNR1 (0.62) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL1829124 0.72 CNR1 (0.76) CNR1CNR2CYP2D6CYP2C9KCNH2
SCHEMBL3524162 0.71 CNR1 (0.60) CNR1CNR2FDFT1
SCHEMBL6515732 0.71 CNR1 (0.55) CNR1CNR2
SCHEMBL3079318 0.69 CNR1 (1.00) CNR1CNR2
SCHEMBL1898233 0.69 CNR1 (1.00) CNR1CNR2
SCHEMBL13894033 0.69 CNR1 (1.00) CNR1CNR2
SCHEMBL13114227 0.69 CNR1 (1.00) CNR1CNR2
SCHEMBL3525559 0.68 FDFT1 (0.59) CNR1CNR2FDFT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001472-A2 GLUCAGON RECEPTOR ANTAGONIST COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE Merck and Co., Inc. (US) 2008-12-17 EP disclosed
WO-2007111864-A2 GLUCAGON RECEPTOR ANTAGONIST COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 2007-10-04 WO disclosed