SCHEMBL2656738

SCHEMBL2656738

Cc1cnc(NC(=O)c2cc(Oc3ccc(C(=O)N4CCC4)nc3)cc(OC3CCN(C4CC4)C3=O)c2)cn1

nearest known ligand 0.63

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GCK P35557 15/20 0.63
KCNH2 Q12809 6/20 0.63
HRH3 Q9Y5N1 5/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2072767 1.00 GCK (0.63) GCKKCNH2HRH3
SCHEMBL2075677 1.00 GCK (0.63) GCKKCNH2HRH3
SCHEMBL2072169 0.98 GCK (0.62) GCKKCNH2HRH3
SCHEMBL2075054 0.98 GCK (0.62) GCKKCNH2HRH3
SCHEMBL2073999 0.98 GCK (0.62) GCKKCNH2HRH3
SCHEMBL2075151 0.91 GCK (0.65) GCKKCNH2HRH3
SCHEMBL2074382 0.91 GCK (0.65) GCKKCNH2HRH3
SCHEMBL2657666 0.91 GCK (0.65) GCKKCNH2HRH3
SCHEMBL2074563 0.89 GCK (0.65) GCKKCNH2HRH3
SCHEMBL2072486 0.89 GCK (0.65) GCKKCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2086964-A2 BENZOYL AMINO HETEROCYCLYL COMPOUNDS USEFUL IN THE TREATMENT OF A DISEASE MEDIATED THROUGH GLK Astra Zeneca AB (SE) 2009-08-12 EP claimed
WO-2008050101-A2 BENZOYL AMINO HETEROCYCLYL COMPOUNDS USEFUL IN THE TREATMENT OF A DISEASE MEDIATED THROUGH GLK ASTRAZENECA AB (SE) 2008-05-02 WO claimed
EP-2086964-A2 BENZOYL AMINO HETEROCYCLYL COMPOUNDS USEFUL IN THE TREATMENT OF A DISEASE MEDIATED THROUGH GLK Astra Zeneca AB (SE) 2009-08-12 EP disclosed
WO-2008050101-A2 BENZOYL AMINO HETEROCYCLYL COMPOUNDS USEFUL IN THE TREATMENT OF A DISEASE MEDIATED THROUGH GLK ASTRAZENECA AB (SE) 2008-05-02 WO disclosed