SCHEMBL2659249

SCHEMBL2659249

C=CC(C)(N)/C=C/c1cccc(C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
PTGS1 P23219 3/20 0.45
PTGS2 P35354 3/20 0.45
ALOX5 P09917 1/20 0.45
RELA Q04206 1/20 0.44
FBP1 P09467 1/20 0.44
NPC1 O15118 1/20 0.43
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
CYP2C19 P33261 1/20 0.38
ACHE P22303 1/20 0.37
NFE2L2 Q16236 2/20 0.36
PIM1 P11309 1/20 0.36
PIM2 Q9P1W9 1/20 0.36
NR1H3 Q13133 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12228136 0.77 TDP1 (0.53) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL29093181 0.76 TDP1 (0.53) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL28448128 0.76 TDP1 (0.53) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL23992499 0.76 TP53 (0.63) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL8542738 0.76 TP53 (0.63) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL8542737 0.76 TP53 (0.63) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL1795132 0.74 PTGS1 (0.69) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL21847980 0.74 PTGS1 (0.69) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL1795130 0.74 PTGS1 (0.69) TP53TDP1PTGS1PTGS2ALOX5
SCHEMBL2091761 0.71 TP53 (0.61) TP53TDP1PTGS1PTGS2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406620-B1 VINYL PHENYL DERIVATIVES AS GLK ACTIVATORS ASTRAZENECA AB (SE) 2006-11-02 EP disclosed