SCHEMBL2662299

SCHEMBL2662299

COC(=O)c1cc(Oc2cnc(C(=O)N(C)C)cn2)cc(OC(C)COC(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GCK P35557 20/20 0.55
RARG P13631 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1040935 1.00 GCK (0.55) GCKRARG
SCHEMBL1043884 0.91 GCK (0.54) GCKRARG
SCHEMBL2086782 0.91 GCK (0.65) GCKRARG
SCHEMBL1040920 0.88 GCK (0.54) GCK
SCHEMBL1040072 0.87 GCK (0.55) GCKRARG
SCHEMBL1043065 0.87 GCK (0.55) GCKRARG
SCHEMBL1043189 0.84 GCK (0.53) GCKRARG
SCHEMBL1042657 0.84 GCK (0.64) GCKRARG
SCHEMBL1427151 0.84 GCK (0.64) GCK
SCHEMBL1041338 0.82 GCK (0.61) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078000-A1 BENZOYL AMINO HETEROCYCLYL COMPOUNDS AS GLUCOKINASE (GLK) ACTIVATORS AstraZeneca AB (SE) 2009-07-15 EP disclosed
WO-2008050117-A1 BENZOYL AMINO HETEROCYCLYL COMPOUNDS AS GLUCOKINASE (GLK) ACTIVATORS ASTRAZENECA AB (SE) 2008-05-02 WO disclosed