SCHEMBL26633045

SCHEMBL26633045

COc1nc(N)c(C#N)c(-c2cccc(-n3ccnc3)c2)c1C#N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 3/20 0.50
ADORA2A P29274 2/20 0.50
KDM4E B2RXH2 7/20 0.49
RXFP1 Q9HBX9 4/20 0.49
NPSR1 Q6W5P4 3/20 0.49
MAPT P10636 2/20 0.49
HSD17B10 Q99714 2/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
CASP1 P29466 1/20 0.49
CASP7 P55210 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
DYRK1A Q13627 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
CYP1A2 P05177 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31215443 1.00 ADORA1 (0.50) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL7017756 0.88 ADORA1 (0.55) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL31215453 0.88 ADORA1 (0.55) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL8928275 0.80 CYP3A4 (0.49) KDM4EHSD17B10MEN1ALDH1A1KMT2A
SCHEMBL26632999 0.77 ADORA2A (0.60) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL7019095 0.77 ADORA1 (0.60) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL28383673 0.75 KDM4E (0.66) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL7023837 0.73 ADORA1 (0.56) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL7016113 0.73 ADORA1 (0.55) ADORA1ADORA2AKDM4ERXFP1NPSR1
SCHEMBL31215452 0.72 ADORA1 (0.54) ADORA1ADORA2AKDM4ERXFP1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023213761-A1 ADENOSINE 2A RECEPTOR MODULATORS FOR USE IN THE TREATMENT OF CANCER UNIVERSITE DE GENEVE (CH) 2023-11-09 WO disclosed