SCHEMBL26640397

SCHEMBL26640397

O=C(O)Cc1ccc(Nc2ncc3c(n2)CNCC3)cc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 4/20 0.47
CDK5R1 Q15078 4/20 0.47
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
GRM5 P41594 1/20 0.45
HTR2C P28335 1/20 0.43
AURKA O14965 1/20 0.42
PDE4B Q07343 5/20 0.41
TYK2 P29597 1/20 0.40
IKBKB O14920 2/20 0.40
PTK2 Q05397 1/20 0.40
SYK P43405 1/20 0.40
EGFR P00533 1/20 0.40
FGFR1 P11362 1/20 0.40
FGFR2 P21802 1/20 0.40
FGFR4 P22455 1/20 0.40
FGFR3 P22607 1/20 0.40
BRD4 O60885 1/20 0.40
PDE4D Q08499 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30648761 0.88 CDK5 (0.46) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL26640913 0.88 CDK5 (0.46) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL26640875 0.87 NEK2 (0.46) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL27054171 0.86 CDK5 (0.49) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL26640775 0.85 CDK2 (0.48) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL26640112 0.85 CDK5 (0.48) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL30648703 0.85 CDK5 (0.48) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL26640174 0.81 CDK5 (0.47) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL30648643 0.81 CDK5 (0.45) CDK5CDK5R1CCNA2CDK2GRM5
SCHEMBL26640389 0.81 CDK5 (0.45) CDK5CDK5R1CCNA2CDK2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023220541-A1 TETRAHYDROPYRIDO[3,4-D]PYRIMIDINES COMPOUNDS AS HPK1 INHIBITORS MERCK PATENT GMBH (DE) 2023-11-16 WO disclosed