SCHEMBL26643045

SCHEMBL26643045

Cc1cnc(-c2nccs2)c(C(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 1/20 0.44
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.35
ALDH1A1 P00352 2/20 0.35
PDPK1 O15530 1/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35
GABRA6 Q16445 1/20 0.35
GABRG1 Q8N1C3 1/20 0.35
GABRG3 Q99928 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Lithium Ion SCHEMBL30644059 0.85 ECE1 (0.36) ECE1KDM4EALDH1A1SMPD3TUBB4A
SCHEMBL26643172 0.84 ECE1 (0.41) ECE1ALDH1A1SMPD3KMT2ATUBB4A
SCHEMBL26769899 0.77 CHRM4 (0.40) KDM4EPDPK1SMPD3RECQL
SCHEMBL30775033 0.76 CSNK2A1 (0.45) ECE1ALDH1A1CSNK2A1TUBB4ATUBB
SCHEMBL16277587 0.76 CSNK2A1 (0.45) ECE1ALDH1A1CSNK2A1TUBB4ATUBB
SCHEMBL29912244 0.74 KDM4E (0.43) KDM4EALDH1A1GABRPGABRDGABRA1
SCHEMBL16114807 0.74 KDM4E (0.43) KDM4EALDH1A1GABRPGABRDGABRA1
SCHEMBL17793760 0.73 KDM4E (0.65) ECE1KDM4ECYP1A2ALDH1A1PDPK1
SCHEMBL25544916 0.73 PIK3C3 (0.44) ECE1KDM4EPDPK1SMPD3KMT2A
SCHEMBL7939469 0.70 HCRTR2 (0.58) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023218023-A1 THIAZOLOARYL-METHYL SUBSTITUTED CYCLIC HYDRAZINE-N-CARBOXAMIDE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2023-11-16 WO disclosed