SCHEMBL2665320

SCHEMBL2665320

CC(C)Oc1cc(OCC(=O)O)cc(C(=O)NC2=NCCS2)c1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 13/20 0.66
RAB9A P51151 12/20 0.66
SMN1; SMN2 Q16637 11/20 0.66
ALDH1A1 P00352 4/20 0.66
KDM4E B2RXH2 2/20 0.66
NFKB1 P19838 1/20 0.64
NFKB2 Q00653 1/20 0.64
RELA Q04206 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.53
LMNA P02545 1/20 0.52
TP53 P04637 2/20 0.51
TOP1 P11387 1/20 0.49
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2665302 0.91 NPC1 (0.65) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13071759 0.86 NPC1 (0.67) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL12652275 0.85 NPC1 (0.57) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13071804 0.83 NPC1 (0.73) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13888123 0.83 NPC1 (0.69) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13888140 0.81 NPC1 (0.63) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13888121 0.81 NPC1 (0.69) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL9071518 0.79 NPC1 (0.64) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13988997 0.78 NPC1 (0.72) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E
SCHEMBL13282846 0.78 NPC1 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7390908-B2 Such as 2-[3,5-Di(2-chlorobenzyloxy)benzoyl)amino]-thiazole; for treatment of diabetes ASTRAZENECA AB (SE) 2008-06-24 US disclosed