SCHEMBL2666464

SCHEMBL2666464

C=C(Cc1cc(OCc2ccccc2F)cc(C(=C)O)c1)Cc1cc(C)on1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCK P35557 2/20 0.38
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38
RARG P13631 1/20 0.38
MAOB P27338 6/20 0.38
HPD P32754 1/20 0.38
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HDAC6 Q9UBN7 3/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC5 Q9UQL6 2/20 0.36
PARP15 Q460N3 1/20 0.35
PARP14 Q460N5 1/20 0.35
PARP10 Q53GL7 1/20 0.35
S1PR1 P21453 1/20 0.35
CASP3 P42574 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649575 0.79 GCK (0.46) GCKRARARARBRARGMAOB
SCHEMBL2666412 0.77 MAOB (0.46) GCKRARARARBRARGMAOB
SCHEMBL2651135 0.76 MAOB (0.41) GCKRARARARBRARGMAOB
SCHEMBL5419201 0.70 GCK (0.68) GCKRARARARBRARG
SCHEMBL2649577 0.70 PARP15 (0.44) GCKRARARARBRARGMAOB
SCHEMBL13703995 0.69 GCK (0.55) GCKRARARARBRARGMAOB
SCHEMBL5421905 0.68 GCK (0.58) GCKRARARARBRARGNPC1
SCHEMBL14018644 0.67 MAOB (0.51) GCKRARARARBRARGMAOB
SCHEMBL14505833 0.65 GCK (0.56) GCKRARARARBRARGMAOB
SCHEMBL2664912 0.65 GCK (0.70) GCKRARARARBRARGNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003000267-A1 AMINO NICOTINATE DERIVATIVES AS GLUCOKINASE (GLK) MODULATORS ASTRAZENECA AB (SE) 2003-01-03 WO disclosed