SCHEMBL2667892

SCHEMBL2667892

N=N/C(=N\N)NC(=O)c1ccc(Cc2cc(-c3ccc(OC(F)(F)F)cc3)n(C3CCCCC3)n2)cc1

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCGR P47871 17/20 0.68
GIPR P48546 6/20 0.44
KCNH2 Q12809 2/20 0.37
DDHD2 O94830 1/20 0.37
SLC5A1 P13866 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9071550 0.86 GCGR (0.68) GCGRGIPRDDHD2
SCHEMBL2252133 0.83 GCGR (0.77) GCGRGIPRKCNH2DDHD2SLC5A1
SCHEMBL9071549 0.81 GCGR (1.00) GCGRGIPRKCNH2CYP3A4CYP2C8
SCHEMBL2667424 0.80 GCGR (0.78) GCGRGIPR
SCHEMBL12360076 0.79 GCGR (1.00) GCGRGIPR
SCHEMBL2251280 0.79 GCGR (0.76) GCGRGIPRSLC5A1
SCHEMBL2667516 0.79 GCGR (0.73) GCGRGIPRKCNH2CYP3A4CYP2C8
SCHEMBL2250476 0.77 GCGR (0.66) GCGRGIPRKCNH2DDHD2SLC5A1
SCHEMBL9071592 0.77 GCGR (0.66) GCGRGIPRKCNH2CYP3A4CYP2C8
SCHEMBL2251890 0.75 GCGR (0.63) GCGRGIPRKCNH2DDHD2SLC5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004069158-A2 SUBSTITUTED PYRAZOLES, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF USE MERCK & CO., INC. (US) 2004-08-19 WO disclosed