SCHEMBL2669129

SCHEMBL2669129

CC(C)Oc1cc(Oc2cnc(C(=O)N3CCC3)cn2)cc(C(=O)N(C)c2cc[nH]n2)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GCK P35557 16/20 0.61
CYP1A2 P05177 1/20 0.52
ABCB1 P08183 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C8 P10632 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2B6 P20813 1/20 0.52
CYP2C19 P33261 1/20 0.52
MEN1 O00255 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
KCNH2 Q12809 3/20 0.40
HRH3 Q9Y5N1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1378805 0.85 GCK (0.72) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL14173451 0.83 GCK (0.61) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL9892948 0.82 GCK (0.67) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL1107723 0.82 GCK (0.67) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL1107293 0.81 GCK (0.66) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL1107651 0.80 GCK (0.68) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL12782140 0.77 GCK (0.66) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL1492818 0.76 GCK (0.78) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL1381418 0.74 GCK (0.58) GCKCYP1A2ABCB1CYP3A4CYP2C8
SCHEMBL12811687 0.74 GCK (0.66) GCKCYP1A2ABCB1CYP3A4CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075073-A1 NOVEL CRYSTALLINE COMPOUND USEFUL AS GLK ACTIVATOR ASTRAZENECA AB (SE) 2008-06-26 WO disclosed