SCHEMBL2669441

SCHEMBL2669441

Cc1ccc(NC(=O)c2cc(OC3=CC=C(C(=O)N(C)C)C(F)C3)c3ccoc3c2)nc1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GCK P35557 15/20 0.50
KCNH2 Q12809 1/20 0.43
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL642946 0.78 GCK (0.53) GCKKCNH2NPC1RAB9AKDM4E
SCHEMBL643430 0.72 GCK (0.62) GCKKCNH2NPC1RAB9A
SCHEMBL10253008 0.70 GCK (0.66) GCKKCNH2NPC1RAB9A
SCHEMBL2645161 0.67 GCK (0.59) GCKKCNH2NPC1RAB9AKDM4E
SCHEMBL643580 0.67 GCK (0.53) GCKKCNH2NPC1RAB9AKDM4E
SCHEMBL645243 0.67 GCK (0.81) GCKKCNH2
SCHEMBL644067 0.67 GCK (0.68) GCKKCNH2NPC1RAB9A
SCHEMBL642311 0.66 GCK (0.65) GCKKCNH2NPC1RAB9AKDM4E
SCHEMBL2644001 0.66 GCK (0.60) GCKKCNH2NPC1RAB9A
SCHEMBL643724 0.66 GCK (0.64) GCKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007122482-A1 FUSED PHENYL AMIDO HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF GLUCOKINASE-MEDIATED DISEASES PFIZER PRODUCTS INC. (US) 2007-11-01 WO disclosed