SCHEMBL26697140

SCHEMBL26697140

CC1(C)OB(c2ccc(CNC(=O)Nc3ccccc3)c(F)c2)OC1(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.53
RAB9A P51151 7/20 0.50
NPC1 O15118 5/20 0.50
PKM P14618 1/20 0.47
MAPK1 P28482 1/20 0.47
PDGFRB P09619 2/20 0.47
KDR P35968 2/20 0.47
KMT2A Q03164 6/20 0.46
MEN1 O00255 4/20 0.46
POLB P06746 1/20 0.45
MAOB P27338 1/20 0.45
MAPT P10636 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
TP53 P04637 1/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 1/20 0.40
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA9 Q16790 2/20 0.40
NAMPT P43490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1290116 0.86 ROCK1 (0.54) ROCK1CA1CA2CA9
SCHEMBL29152163 0.85 ROCK1 (0.54) ROCK1NPC1POLBHPGDALDH1A1
SCHEMBL20365272 0.83 ROCK1 (0.54) ROCK1CA1CA2CA9
SCHEMBL28616950 0.81 ROCK1 (0.52) ROCK1RAB9APKMMAPK1KMT2A
SCHEMBL5675802 0.81 NPC1 (0.62) RAB9ANPC1PDGFRBKDRKMT2A
SCHEMBL5678324 0.80 NPC1 (0.51) RAB9ANPC1PDGFRBKDRKMT2A
SCHEMBL20359137 0.80 ROCK1 (0.51) ROCK1CA1CA2CA9
SCHEMBL423204 0.77 PDGFRB (0.61) RAB9ANPC1PDGFRBKDRKMT2A
SCHEMBL1290158 0.77 PRMT5 (0.57) ROCK1CA1CA2CA9
SCHEMBL14898157 0.76 ROCK1 (0.63) ROCK1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117164591-A Pyrrolopyrimidine compound, preparation method and pharmaceutical application thereof 中国医学科学院药物研究所 2023-12-05 CN disclosed
WO-2023226580-A1 PYRROLOPYRIMIDINE COMPOUND, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 中国医学科学院药物研究所 2023-11-30 WO disclosed