SCHEMBL2679102

SCHEMBL2679102

CCN1CCN(Cc2ccc(C(=O)Nc3ccc(C)c(NC(=O)C=Cc4cccnc4)c3)cc2C(F)(F)F)CC1

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 2/20 0.65
KIT P10721 2/20 0.65
EGFR P00533 1/20 0.65
BRAF P15056 1/20 0.65
NR2C2 P49116 3/20 0.64
BTK Q06187 3/20 0.64
HCK P08631 1/20 0.62
GCK P35557 1/20 0.62
HTT P42858 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10054812 1.00 CSF1R (0.65) CSF1RKITEGFRBRAFNR2C2
SCHEMBL10054810 0.94 BRAF (0.74) CSF1RKITEGFRBRAF
SCHEMBL2679098 0.94 BRAF (0.74) CSF1RKITEGFRBRAF
SCHEMBL10054811 0.92 KIT (0.62) CSF1RKITEGFRBRAFNR2C2
SCHEMBL2679279 0.92 KIT (0.62) CSF1RKITEGFRBRAFNR2C2
SCHEMBL2679815 0.92 BTK (0.66) CSF1RKITEGFRBRAFNR2C2
SCHEMBL10054836 0.92 BTK (0.66) CSF1RKITEGFRBRAFNR2C2
SCHEMBL10054815 0.92 BRAF (0.70) CSF1RKITEGFRBRAF
SCHEMBL2679557 0.89 BRAF (0.66) CSF1RKITEGFRBRAFHTT
SCHEMBL10077763 0.89 BRAF (0.66) CSF1RKITEGFRBRAFHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8426446-B2 Acrylamide derivative and use thereof in manufacture of medicament BEIJING SHIQIAO BIOPHARM CO. LTD. (CN) 2013-04-23 US claimed
US-20120116075-A1 Acrylamide Derivative And Use Thereof In Manufacture Of Medicament BEIJING JIASHILIANBO PHARM SCI & TECH CO. LTD 2012-05-10 US claimed
US-8426446-B2 Acrylamide derivative and use thereof in manufacture of medicament BEIJING SHIQIAO BIOPHARM CO. LTD. (CN) 2013-04-23 US disclosed
US-20120116075-A1 Acrylamide Derivative And Use Thereof In Manufacture Of Medicament BEIJING JIASHILIANBO PHARM SCI & TECH CO. LTD 2012-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120116075-A1 Acrylamide Derivative And Use Thereof In Manufacture Of Medicament ABL1, ABL2, BCR CSF1R 2608/4885KIT 399/4885EGFR 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.