SCHEMBL2679153

SCHEMBL2679153

Cc1ccc(NC(=O)c2cccc(C(F)(F)F)c2)cc1NC(=O)C=Cc1cccnc1

nearest known ligand 0.75

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BRAF P15056 10/20 0.75
CSF1R P07333 7/20 0.75
NAMPT P43490 2/20 0.61
KIT P10721 4/20 0.60
PIKFYVE Q9Y2I7 1/20 0.57
KDR P35968 1/20 0.56
MAPK14 Q16539 1/20 0.56
BMX P51813 1/20 0.56
DDR1 Q08345 1/20 0.56
DDR2 Q16832 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10054791 1.00 BRAF (0.75) BRAFCSF1RNAMPTKITPIKFYVE
SCHEMBL10077740 0.93 CSF1R (0.73) BRAFCSF1RNAMPTKITKDR
SCHEMBL2679147 0.93 CSF1R (0.73) BRAFCSF1RNAMPTKITKDR
SCHEMBL10054793 0.93 BRAF (0.63) BRAFCSF1RNAMPTKIT
SCHEMBL2678795 0.93 BRAF (0.63) BRAFCSF1RNAMPTKIT
Bromomethane SCHEMBL2679140 0.90 BRAF (0.59) BRAFCSF1RNAMPTKITPIKFYVE
SCHEMBL2679254 0.90 BRAF (0.59) BRAFCSF1RNAMPT
SCHEMBL10054797 0.90 BRAF (0.59) BRAFCSF1RNAMPT
SCHEMBL2679829 0.89 BRAF (0.58) BRAFCSF1RNAMPTKITKDR
SCHEMBL10054792 0.89 BRAF (0.58) BRAFCSF1RNAMPTKITKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102421754-B Acrylamide derivative and use thereof in manufacture of medicament BEIJING SHIQIAO BIOPHAM CO LTD 2013-11-27 CN claimed
US-8426446-B2 Acrylamide derivative and use thereof in manufacture of medicament BEIJING SHIQIAO BIOPHARM CO. LTD. (CN) 2013-04-23 US claimed
US-20120116075-A1 Acrylamide Derivative And Use Thereof In Manufacture Of Medicament BEIJING JIASHILIANBO PHARM SCI & TECH CO. LTD 2012-05-10 US claimed
CN-102421754-B Acrylamide derivative and use thereof in manufacture of medicament BEIJING SHIQIAO BIOPHAM CO LTD 2013-11-27 CN disclosed
US-8426446-B2 Acrylamide derivative and use thereof in manufacture of medicament BEIJING SHIQIAO BIOPHARM CO. LTD. (CN) 2013-04-23 US disclosed
US-20120116075-A1 Acrylamide Derivative And Use Thereof In Manufacture Of Medicament BEIJING JIASHILIANBO PHARM SCI & TECH CO. LTD 2012-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120116075-A1 Acrylamide Derivative And Use Thereof In Manufacture Of Medicament ABL1, ABL2, BCR BRAF 21/4885CSF1R 2608/4885NAMPT 3700/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.