SCHEMBL26795366

SCHEMBL26795366

CNc1nc2c(cc1N)C(=O)NCC2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.41
PIM1 P11309 3/20 0.39
PIM2 Q9P1W9 3/20 0.39
PARP1 P09874 2/20 0.39
CDC7 O00311 7/20 0.37
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CDK9 P50750 1/20 0.36
PLK1 P53350 1/20 0.36
CCNA1 P78396 1/20 0.36
GRM5 P41594 2/20 0.36
PARP10 Q53GL7 2/20 0.36
PARP11 Q9NR21 1/20 0.36
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.34
MAP4K1 Q92918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31732376 1.00 PDE4B (0.41) PDE4BPIM1PIM2PARP1CDC7
SCHEMBL26660618 0.78 POLB (0.43) PIM1PIM2PARP1GRM5PARP10
SCHEMBL31501903 0.78 POLB (0.43) PIM1PIM2PARP1GRM5PARP10
SCHEMBL26660637 0.71 MAP4K1 (0.45) PARP1GRM5PARP10PARP11CYP1A2
SCHEMBL31501830 0.71 MAP4K1 (0.45) PARP1GRM5PARP10PARP11CYP1A2
SCHEMBL30669000 0.70 PARP10 (0.47) PARP1GRM5PARP10PARP11KDM4E
SCHEMBL26671057 0.70 PARP10 (0.47) PARP1GRM5PARP10PARP11KDM4E
SCHEMBL17111725 0.70 PDE4B (0.46) PDE4BPIM1PIM2PARP1CDC7
SCHEMBL23649631 0.68 GRM5 (0.46) PDE4BPIM1PIM2PARP1CDC7
SCHEMBL20302818 0.68 PARP10 (0.41) PIM1PIM2PARP1CDC7CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023230612-A1 HETEROCYCLIC PAD4 INHIBITORS CELGENE CORPORATION (US) 2023-11-30 WO disclosed