SCHEMBL26943136

SCHEMBL26943136

O=S(=O)(c1ccc(C2CCNCC2)cc1)N1CCC(Nc2ncc(C(F)(F)F)c(O[C@H]3CCOC3)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 8/20 0.45
MAPK8 P45983 2/20 0.42
CDK2 P24941 5/20 0.41
CCNE1 P24864 4/20 0.41
CDK1 P06493 3/20 0.41
CCNB1 P14635 3/20 0.41
KDR P35968 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
CHUK O15111 1/20 0.40
MAPK9 P45984 1/20 0.40
MAPK10 P53779 1/20 0.40
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
CCNT1 O60563 2/20 0.40
CDK4 P11802 2/20 0.40
CCND1 P24385 2/20 0.40
CCND3 P30281 2/20 0.40
CDK7 P50613 2/20 0.40
CDK9 P50750 2/20 0.40
CCNH P51946 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26943388 0.95 IKBKB (0.42) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26943389 0.95 IKBKB (0.42) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26943303 0.95 IKBKB (0.42) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26943137 0.93 CDK2 (0.41) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL29763125 0.92 CDK2 (0.41) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26919483 0.92 CDK2 (0.41) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26919480 0.92 CDK2 (0.41) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26943236 0.92 IKBKB (0.47) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26943302 0.89 IKBKB (0.45) IKBKBMAPK8CDK2CCNE1CDK1
SCHEMBL26946820 0.89 IKBKB (0.41) IKBKBMAPK8CDK2CCNE1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4289835-A1 CDK INHIBITOR Shanghai Qilu Pharmaceutical Research and Development Centre Ltd. (CN) 2023-12-13 EP disclosed