SCHEMBL27103013

SCHEMBL27103013

C[C@H]1CNCCN1c1ccnc(F)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.44
GSK3B P49841 4/20 0.41
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 1/20 0.41
LATS1 O95835 1/20 0.40
HTR2C P28335 7/20 0.40
HTR2B P41595 5/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CDK4 P11802 2/20 0.39
HTR2A P28223 4/20 0.39
MET P08581 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
HRH4 Q9H3N8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL22836915 0.99 RAD52 (0.46) RAD52GSK3BROCK2ROCK1LATS1
Hydrochloric Acid SCHEMBL22836914 0.99 RAD52 (0.46) RAD52GSK3BROCK2ROCK1LATS1
Hydrochloric Acid SCHEMBL30062597 0.99 RAD52 (0.46) RAD52GSK3BROCK2ROCK1LATS1
Hydrochloric Acid SCHEMBL30063113 0.99 RAD52 (0.46) RAD52GSK3BROCK2ROCK1LATS1
SCHEMBL21098363 0.81 GSK3B (0.42) RAD52GSK3BROCK2ROCK1LATS1
SCHEMBL21098364 0.81 GSK3B (0.42) RAD52GSK3BROCK2ROCK1LATS1
SCHEMBL5461889 0.79 GSK3B (0.52) RAD52GSK3BROCK1LATS1HTR2C
SCHEMBL26669231 0.79 GSK3B (0.52) RAD52GSK3BROCK1LATS1HTR2C
SCHEMBL38663101 0.79 GSK3B (0.52) RAD52GSK3BROCK1LATS1HTR2C
SCHEMBL5630952 0.78 RAD52 (0.49) RAD52GSK3BROCK2LATS1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3990442-B1 RHO KINASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION INC (US) 2024-02-28 EP disclosed