SCHEMBL2726041

SCHEMBL2726041

O=CCc1ccc(-c2ccc3c(N4CCOCC4)nc(Cl)nc3c2)o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.46
PIK3CA P42336 1/20 0.38
PRKDC P78527 6/20 0.38
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
GAA P10253 2/20 0.37
GLA P06280 1/20 0.37
HPGD P15428 1/20 0.37
PI4KB Q9UBF8 1/20 0.36
MTOR P42345 1/20 0.36
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAK O14976 1/20 0.36
EGLN1 Q9GZT9 2/20 0.35
MAT2A P31153 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HRH1 P35367 1/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2731944 0.86 SMN1; SMN2 (0.51) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL8408289 0.86 PI4KB (0.48) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL2727144 0.85 SMN1; SMN2 (0.47) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL2726605 0.84 SMN1; SMN2 (0.47) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL8408288 0.84 SMN1; SMN2 (0.48) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL2726476 0.82 SMN1; SMN2 (0.53) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL2726036 0.80 SMN1; SMN2 (0.51) SMN1; SMN2PIK3CAPRKDCALDH1A1GAA
SCHEMBL8408337 0.79 SMN1; SMN2 (0.47) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL8408334 0.79 SMN1; SMN2 (0.58) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1
SCHEMBL2726335 0.79 SMN1; SMN2 (0.47) SMN1; SMN2PIK3CAPRKDCKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058671-A1 SUBSTITUTED QUINAZOLINE AND PYRIDO-PYRIMIDINE DERIVATIVES ENDO PHARMACEUTICALS INC. (US) 2012-05-03 WO disclosed