SCHEMBL2726162

SCHEMBL2726162

Cc1csc([C@H]2CCCN2C(=O)c2cc(-c3ccn(C)n3)nc(-c3nnc([C@@](C)(Cc4ccccc4)NC(=O)O)o3)c2)n1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.36
TRPV1 Q8NER1 2/20 0.35
KCNK3 O14649 1/20 0.34
POLB P06746 1/20 0.34
CPT1A P50416 6/20 0.33
NAA50 Q9GZZ1 1/20 0.33
CPT2 P23786 4/20 0.32
AADAT Q8N5Z0 3/20 0.32
PKM P14618 1/20 0.31
CPT1B Q92523 1/20 0.31
CPS1 P31327 1/20 0.31
JMJD6 Q6NYC1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2728191 0.92 SMN1; SMN2 (0.38) SMN1; SMN2TRPV1POLBCPT1ANAA50
SCHEMBL2727033 0.91 SMN1; SMN2 (0.37) SMN1; SMN2TRPV1POLBCPT1ANAA50
SCHEMBL2725792 0.91 BACE1 (0.35) SMN1; SMN2TRPV1KCNK3POLBCPT1A
SCHEMBL2725793 0.91 BACE1 (0.35) SMN1; SMN2TRPV1KCNK3POLBCPT1A
SCHEMBL2727845 0.90 CPT1A (0.39) SMN1; SMN2TRPV1POLBCPT1ACPT2
SCHEMBL2726866 0.90 SMN1; SMN2 (0.37) SMN1; SMN2TRPV1POLBCPT1ANAA50
SCHEMBL2726697 0.90 TRPV1 (0.36) SMN1; SMN2TRPV1POLBCPT1ANAA50
SCHEMBL2726726 0.90 SMN1; SMN2 (0.37) SMN1; SMN2TRPV1POLBCPT1ANAA50
SCHEMBL2731961 0.90 SMN1; SMN2 (0.37) SMN1; SMN2TRPV1POLBCPT1ANAA50
SCHEMBL2727730 0.89 CPT1A (0.34) SMN1; SMN2TRPV1KCNK3CPT1ANAA50

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed