SCHEMBL27264104

SCHEMBL27264104

COc1cc(F)c(F)cc1I

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.41
HTR2C P28335 7/20 0.41
HTR2B P41595 6/20 0.41
HTR1A P08908 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
PMP22 Q01453 2/20 0.40
LMNA P02545 2/20 0.40
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
TUBB1 Q9H4B7 2/20 0.34
MAPT P10636 1/20 0.33
HRH1 P35367 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22025397 0.88 HTR2A (0.40) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL22342696 0.88 HTR2A (0.44) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL22342695 0.84 HTR2A (0.38) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL31401783 0.82 NPC1 (0.41) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL16664687 0.82 HTR2A (0.41) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL19703128 0.82 HTR2A (0.44) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL31021971 0.82 HTR2A (0.41) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL16290528 0.82 MAPT (0.44) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL29888847 0.82 MAPT (0.44) HTR2AHTR2CHTR2BHTR1ACYP3A4
SCHEMBL2111831 0.82 HTR2A (0.41) HTR2AHTR2CHTR2BHTR1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024015412-A1 TETRAHYDRONAPHTHALENE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2024-01-18 WO disclosed