SCHEMBL27280642

SCHEMBL27280642

Cc1cc(F)c(-c2cc(Nc3cnc(C#N)cn3)n[nH]2)c(O[C@@H]2CCC[C@H]2N)c1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 20/20 0.55
KCNH2 Q12809 13/20 0.55
NUAK1 O60285 1/20 0.47
CHEK2 O96017 1/20 0.47
RPS6KB1 P23443 1/20 0.47
FLT3 P36888 1/20 0.47
BLK P51451 1/20 0.47
PRKAG1 P54619 1/20 0.47
PRKAA1 Q13131 1/20 0.47
PRKAB1 Q9Y478 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30954374 1.00 CHEK1 (0.55) CHEK1KCNH2NUAK1CHEK2RPS6KB1
SCHEMBL27280726 0.89 CHEK1 (0.52) CHEK1KCNH2NUAK1CHEK2RPS6KB1
SCHEMBL24977540 0.88 CHEK1 (0.54) CHEK1KCNH2NUAK1CHEK2RPS6KB1
SCHEMBL30106185 0.88 CHEK1 (0.54) CHEK1KCNH2NUAK1CHEK2RPS6KB1
SCHEMBL24977886 0.88 CHEK1 (0.54) CHEK1KCNH2NUAK1CHEK2RPS6KB1
SCHEMBL30106213 0.88 CHEK1 (0.54) CHEK1KCNH2NUAK1CHEK2RPS6KB1
SCHEMBL27280618 0.87 CHEK1 (0.58) CHEK1KCNH2
SCHEMBL27312354 0.87 CHEK1 (0.57) CHEK1KCNH2
SCHEMBL27312710 0.87 CHEK1 (0.57) CHEK1KCNH2
SCHEMBL27312343 0.87 CHEK1 (0.57) CHEK1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024118564-A1 CHECKPOINT KINASE 1 (CHK1) INHIBITORS AND USES THEREOF BOUNDLESS BIO, INC. (US) 2024-06-06 WO disclosed