SCHEMBL27282452

SCHEMBL27282452

[CH2]CCNC(=O)c1cc(NC(=O)c2cc([N+](=O)[O-])cn2C)cn1C

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRAS P01112 9/20 0.47
ESR1 P03372 9/20 0.47
ESR2 Q92731 9/20 0.47
TOP1 P11387 2/20 0.47
POLB P06746 2/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
HIF1A Q16665 1/20 0.47
AR P10275 1/20 0.39
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HPSE Q9Y251 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
NAMPT P43490 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27272956 1.00 HRAS (0.47) HRASESR1ESR2TOP1POLB
SCHEMBL27275434 1.00 HRAS (0.47) HRASESR1ESR2TOP1POLB
SCHEMBL27279001 1.00 HRAS (0.47) HRASESR1ESR2TOP1POLB
SCHEMBL27276235 1.00 HRAS (0.47) HRASESR1ESR2TOP1POLB
SCHEMBL27281880 0.93 TOP1 (0.43) HRASESR1ESR2TOP1POLB
SCHEMBL26374814 0.87 HRAS (0.47) HRASESR1ESR2TOP1POLB
SCHEMBL6257041 0.85 HRAS (0.47) HRASESR1ESR2TOP1POLB
SCHEMBL30644155 0.85 HRAS (0.47) HRASESR1ESR2TOP1POLB
Hydrochloric Acid SCHEMBL6178124 0.85 TOP1 (0.55) HRASESR1ESR2TOP1POLB
SCHEMBL1844965 0.84 HDAC1 (0.51) HRASESR1ESR2TOP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1018825-B Process for preparing poly-4-aminopyrrole-2-carboxamido derivatives ERBA FARMITALIA (IT) 1992-10-28 CN disclosed