SCHEMBL2729359

SCHEMBL2729359

CC(C)(C)N1CCN(CCc2ccc3c(c2I)COC3=O)CC1

nearest known ligand 0.62

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 17/20 0.62
KCNH2 Q12809 11/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2732990 0.82 KCNJ1 (0.60) KCNJ1KCNH2
SCHEMBL2731889 0.82 KCNH2 (0.55) KCNJ1KCNH2
Hydrochloric Acid SCHEMBL2733934 0.81 KCNJ1 (0.58) KCNJ1KCNH2
SCHEMBL2733631 0.78 KCNJ1 (0.49) KCNJ1KCNH2
SCHEMBL10234057 0.77 KCNJ1 (1.00) KCNJ1KCNH2
SCHEMBL2729938 0.73 KCNJ1 (0.46) KCNJ1KCNH2
Trifluoroacetic Acid SCHEMBL17360760 0.71 KCNJ1 (0.80) KCNJ1KCNH2
SCHEMBL14782785 0.71 KCNJ1 (0.85) KCNJ1KCNH2
SCHEMBL15210266 0.71 KCNJ1 (0.83) KCNJ1KCNH2
SCHEMBL296919 0.70 KCNJ1 (0.83) KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632464-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058134-A1 INHIBITORS OF THE RENAL OUTER MEDULLARY POTASSIUM CHANNEL MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed