SCHEMBL27311528

SCHEMBL27311528

Cc1ccccc1C(=O)Nc1ccc(C(=O)N2c3ccccc3C(N(C)C)CC2C)cc1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 6/20 0.66
AVPR2 P30518 5/20 0.66
AVPR1B P47901 2/20 0.66
OXTR P30559 2/20 0.66
ABCB11 O95342 1/20 0.66
HTR1A P08908 1/20 0.66
CHRM1 P11229 1/20 0.66
SLC6A4 P31645 1/20 0.66
ADRA1A P35348 1/20 0.66
OPRM1 P35372 1/20 0.66
PTGDR2 Q9Y5Y4 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712149 0.91 AVPR1A (0.70) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8713010 0.85 AVPR1A (0.70) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8715943 0.85 AVPR1A (0.69) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8712963 0.85 AVPR1A (0.69) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8718080 0.83 AVPR1A (0.73) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL27323365 0.83 PTGDR2 (0.55) PTGDR2
SCHEMBL8712791 0.83 AVPR1A (0.67) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8715795 0.82 AVPR1A (0.71) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8712361 0.81 AVPR1A (0.70) AVPR1AAVPR2AVPR1BOXTRABCB11
SCHEMBL8714659 0.81 AVPR1A (0.57) AVPR1AAVPR2AVPR1BOXTRABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1048484-C A process for preparing a composition containing benzoheterocycles OTSUKA PHARMA CO LTD (JP) 2000-01-19 CN disclosed
CN-1027505-C Process for preparing benzoheterocyclic compounds OTSUKA PHARMA CO LTD (JP) 1995-01-25 CN disclosed