SCHEMBL27320171

SCHEMBL27320171

CC(C)C[C@H](N)CS(=O)(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 5/20 0.42
ERAP1 Q9NZ08 2/20 0.42
ERAP2 Q6P179 1/20 0.42
TSHR P16473 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
NFKB1 P19838 1/20 0.41
THPO P40225 1/20 0.41
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
PMP22 Q01453 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
SLC7A5 Q01650 1/20 0.39
SLC1A3 P43003 2/20 0.39
SLC1A2 P43004 2/20 0.39
LAP3 P28838 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6034381 1.00 ANPEP (0.42) ANPEPERAP1ERAP2TSHRCYP3A4
SCHEMBL27422167 1.00 ANPEP (0.42) ANPEPERAP1ERAP2TSHRCYP3A4
SCHEMBL30589985 0.78 ANPEP (0.44) ANPEPERAP1ERAP2TSHRCYP3A4
SCHEMBL9294910 0.78 SLC22A6 (0.36) LMNASLC22A6
SCHEMBL28794128 0.78 SLC22A6 (0.36) LMNASLC22A6
SCHEMBL15980620 0.78 ANPEP (0.44) ANPEPERAP1ERAP2TSHRCYP3A4
SCHEMBL356000 0.77 S1PR2 (0.41) ANPEPERAP1ERAP2TSHRCYP3A4
SCHEMBL354858 0.77 S1PR2 (0.41) ANPEPERAP1ERAP2TSHRCYP3A4
SCHEMBL355325 0.77 S1PR2 (0.41) ANPEPERAP1ERAP2TSHRCYP3A4
Isopropylamine SCHEMBL27887484 0.77 SLC22A6 (0.39) ANPEPERAP1TSHRLMNASLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1046512-C Novel mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase and ace MERRELL DOW PHARMA (US) 1999-11-17 CN claimed
CN-1069317-C Novel indane-2-mercaptoacetylamide disulfide derivs. useful as inhibitors of enkephalinase MERRELL PHARMA INC (US) 2001-08-08 CN disclosed
CN-1046512-C Novel mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase and ace MERRELL DOW PHARMA (US) 1999-11-17 CN disclosed
CN-1142826-A Novel mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase and ace MERRELL DOW PHARMA (US) 1997-02-12 CN disclosed
CN-1142831-A Novel 2-substituted indane-2-mercaploacetylamide disulfide derivatives useful as inhibitors of enkephalinase and ace MERRELL DOW PHARMA (US) 1997-02-12 CN disclosed
CN-1140451-A Novel 1, 2-indan-2-mercaptoacetamide disulfide derivatives as enkephalinase inhibitors MERRELL DOW PHARMA (US) 1997-01-15 CN disclosed