SCHEMBL2733825

SCHEMBL2733825

N#Cc1ccnc(N2CCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCC3(CCCN(Cc4c[nH]c5ccccc45)C3=O)CC2)c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 20/20 0.67
HCRTR1 O43613 15/20 0.67
HTR1A P08908 1/20 0.58
TSPO P30536 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2131984 0.97 HCRTR2 (0.71) HCRTR2HCRTR1HTR1ATSPO
SCHEMBL9949316 0.93 HCRTR2 (0.64) HCRTR2HCRTR1HTR1ATSPO
SCHEMBL6422588 0.86 HCRTR2 (0.75) HCRTR2HCRTR1HTR1ATSPO
SCHEMBL2132317 0.84 HCRTR2 (0.70) HCRTR2HCRTR1
SCHEMBL2133390 0.84 HCRTR2 (0.75) HCRTR2HCRTR1HTR1ATSPO
SCHEMBL2133507 0.84 HCRTR2 (0.73) HCRTR2HCRTR1HTR1ATSPO
SCHEMBL2605432 0.81 HCRTR2 (0.57) HCRTR2HCRTR1
SCHEMBL2132759 0.80 HCRTR2 (0.77) HCRTR2HCRTR1HTR1ATSPO
SCHEMBL2027169 0.80 HCRTR2 (1.00) HCRTR2HCRTR1
SCHEMBL2134028 0.80 HCRTR2 (0.71) HCRTR2HCRTR1HTR1ATSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632924-A1 DIAZA-SPIRO[5.5]UNDECANES USEFUL AS OREXIN RECEPTOR ANTAGONISTS Novartis AG (CH) 2013-09-04 EP disclosed
WO-2012055888-A1 DIAZA-SPIRO[5.5]UNDECANES USEFUL AS OREXIN RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2012-05-03 WO disclosed