SCHEMBL2734533

SCHEMBL2734533

CC(C)(C)N1CCCC(n2cc(-c3ccc4c(c3)c(-c3ccncc3)nn4C(c3ccccc3)(c3ccccc3)c3ccccc3)cn2)C1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.34
BTK Q06187 10/20 0.34
TYRO3 Q06418 1/20 0.32
ALK Q9UM73 4/20 0.31
RIPK1 Q13546 1/20 0.31
SOS1 Q07889 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2733119 0.85 BTK (0.44) BTK
SCHEMBL15248283 0.71 FGFR3 (0.46) BTK
SCHEMBL16025986 0.69 AXL (0.42) DRD2TYRO3ALK
SCHEMBL16025543 0.68 AXL (0.41) DRD2ALK
SCHEMBL16025985 0.67 LRRK2 (0.49)
SCHEMBL30084116 0.67 PTGER1 (0.38) BTK
SCHEMBL30084130 0.67 PTGER1 (0.38)
SCHEMBL173515 0.67 PTGER1 (0.38) BTK
SCHEMBL2732363 0.67 DCLK1 (0.40)
SCHEMBL2733380 0.67 MKNK1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2632268-A2 NOVEL COMPOUNDS THAT ARE ERK INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-09-04 EP disclosed
WO-2012058127-A2 NOVEL COMPOUNDS THAT ARE ERK INHIBITORS SCHERING CORPORATION (US) 2012-05-03 WO disclosed