SCHEMBL27360352

SCHEMBL27360352

C/C(=C/N[C@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](CO)c1ccc(-c2ccncc2)cc1)C(C)C)N=N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.39
MLX Q9UH92 1/20 0.39
PREP P48147 1/20 0.39
ELANE P08246 9/20 0.38
ROCK2 O75116 6/20 0.36
MAPK13 O15264 1/20 0.36
RPS6KA5 O75582 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
PRKCG P05129 1/20 0.36
CDK1 P06493 1/20 0.36
PRKACA P17612 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CDK2 P24941 1/20 0.36
MAPK1 P28482 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
CLK2 P49760 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27360354 0.93 ELANE (0.39) XIAPMLXELANETAAR1SLC6A2
SCHEMBL27360356 0.92 XIAP (0.37) XIAPMLXELANETAAR1SLC6A2
SCHEMBL27360246 0.92 ELANE (0.40) XIAPMLXPREPELANEROCK2
SCHEMBL27360367 0.91 XIAP (0.38) XIAPMLXPREPELANETAAR1
SCHEMBL27360361 0.91 MAPK1 (0.38) XIAPMLXPREPELANEMAPK1
SCHEMBL27360359 0.91 XIAP (0.37) XIAPMLXPREPELANETAAR1
SCHEMBL27360362 0.91 ELANE (0.40) XIAPMLXELANETAAR1
SCHEMBL27360580 0.90 XIAP (0.38) XIAPMLXPREPELANETAAR1
SCHEMBL27360364 0.90 ELANE (0.37) XIAPMLXPREPELANEGSK3B
SCHEMBL27360245 0.89 ELANE (0.41) XIAPMLXELANETAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024040080-A1 KRAS INHIBITOR CONJUGATES ERASCA, INC. (US) 2024-02-22 WO disclosed