SCHEMBL27361537

SCHEMBL27361537

CSc1ncc(Br)c(NC(C)C)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 14/20 0.46
KDR P35968 13/20 0.46
CDK2 P24941 13/20 0.46
CDK7 P50613 3/20 0.40
CDK9 P50750 3/20 0.40
IGF1R P08069 2/20 0.40
CHEK1 O14757 1/20 0.40
AURKA O14965 1/20 0.40
DAPK3 O43293 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
LCK P06239 1/20 0.40
FYN P06241 1/20 0.40
CSF1R P07333 1/20 0.40
RET P07949 1/20 0.40
PDGFRB P09619 1/20 0.40
FGFR1 P11362 1/20 0.40
LTK P29376 1/20 0.40
GRK5 P34947 1/20 0.40
MAPK8 P45983 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29991317 1.00 CDK1 (0.46) CDK1KDRCDK2CDK7CDK9
SCHEMBL27225058 0.82 IGF1R (0.34) CDK1KDRCDK2CDK7CDK9
SCHEMBL10998952 0.80 KDM4E (0.35) CDK1KDRCDK2IGF1RCA2
SCHEMBL28300418 0.80 KDM4E (0.42) CDK1CDK2IGF1RLRRK2CCNB1
SCHEMBL29533105 0.80 KDM4E (0.35) CDK1KDRCDK2IGF1RCA2
SCHEMBL22200723 0.79 APP (0.35) CDK2MAPK8MAPK9GSK3BKDM4E
SCHEMBL6416479 0.79 KDM4E (0.35) CDK1CDK2IGF1RCCNB1CCNE1
SCHEMBL25211340 0.78 NTRK1 (0.35) LMNAHTTSMN1; SMN2KDM4EMEN1
SCHEMBL5067063 0.77 MEN1 (0.34) CDK1KDRCDK2CA2LMNA
SCHEMBL15357782 0.77 KDR (0.47) CDK1KDRCDK2CDK7CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024039903-A2 CDK2 INHIBITORS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2024-02-22 WO disclosed