SCHEMBL27365315

SCHEMBL27365315

COC(=O)c1ccc(C#CC2CCCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 2/20 0.51
FFAR4 Q5NUL3 2/20 0.51
PTPN11 Q06124 1/20 0.49
CYP2C19 P33261 2/20 0.48
MEN1 O00255 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
KMT2A Q03164 1/20 0.48
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
EPHX2 P34913 1/20 0.47
MAPT P10636 2/20 0.45
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
CA12 O43570 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27363242 0.98 FFAR1 (0.52) FFAR1FFAR4PTPN11CYP2C19MEN1
SCHEMBL13757141 0.94 PTPN11 (0.51) FFAR1FFAR4PTPN11NPC1ALDH1A1
SCHEMBL22197977 0.87 PTPN11 (0.46) FFAR1FFAR4PTPN11NPC1ALDH1A1
SCHEMBL3007588 0.87 PTPN11 (0.46) PTPN11CYP2C19MEN1CYP1A2CYP2D6
SCHEMBL13831561 0.84 FFAR1 (0.45) FFAR1FFAR4PTPN11MEN1KMT2A
SCHEMBL17996034 0.84 FFAR1 (0.51) FFAR1FFAR4CYP2C19CYP1A2CYP2C9
SCHEMBL14715015 0.83 PTPN11 (0.48) PTPN11NPC1ALDH1A1SMN1; SMN2MAPT
SCHEMBL3018699 0.82 PTPN11 (0.47) PTPN11NPC1ALDH1A1SMN1; SMN2MAPT
SCHEMBL3587230 0.81 FFAR1 (0.43) FFAR1FFAR4ALDH1A1MAPTHAO1
SCHEMBL4498928 0.80 FFAR1 (0.60) FFAR1FFAR4PTPN11KMT2AHAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024054624-A1 MODULATORS OF ALPHA-1 ANTITRYPSIN VERTEX PHARMACEUTICALS INCORPORATED (US) 2024-03-14 WO disclosed