Pyrazinoic Acid

Pyrazinoic Acid

SCHEMBL27366676

O=C(O)c1cnccn1.[NaH].[NaH].[NaH]

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.95
NAPRT Q6XQN6 2/20 0.95
HCAR2 Q8TDS4 1/20 0.95
TSHR P16473 2/20 0.68
ADORA3 P0DMS8 1/20 0.68
MC4R P32245 1/20 0.68
ADRA1A P35348 1/20 0.68
MC3R P41968 1/20 0.68
BAZ2B Q9UIF8 1/20 0.50
LMNA P02545 2/20 0.46
P4HTM Q9NXG6 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MAPT P10636 2/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 2/20 0.44
ALOX15 P16050 1/20 0.44
KMT2A Q03164 1/20 0.44
KDM6B O15054 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyrazinoic Acid SCHEMBL9478203 1.00 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL28046860 1.00 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL29651929 0.98
Pyrazinoic Acid SCHEMBL23757 0.98
Pyrazinoic Acid SCHEMBL28292273 0.96 KDM4E (0.87) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL10349317 0.95 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL8335237 0.95 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL623119 0.95 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL6631652 0.95 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3
Pyrazinoic Acid SCHEMBL8978502 0.95 KDM4E (0.95) KDM4ENAPRTHCAR2TSHRADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1063180-C 5H, 10H-imidazo [1, 2 -a] indeno [1, 2 -e] pyrazin-4-one derivatives, preparation thereof, and drugs containing said derivatives RHONE POULENC RORER SA (FR) 2001-03-14 CN disclosed
CN-1180357-A 5H, 10H-imidazo [1, 2-a ] indeno [1, 2-e ] pyrazin-4-one derivatives, preparation thereof and medicaments containing same RHONE POULENC RORER SA (FR) 1998-04-29 CN disclosed