SCHEMBL27375976

SCHEMBL27375976

C1CCN(C[C@H]2CCNC2)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.52
ADRA2C P18825 1/20 0.52
SLC6A1 P30531 2/20 0.41
GABRA5 P31644 2/20 0.41
GABRB2 P47870 2/20 0.41
SLC6A12 P48065 2/20 0.41
SLC6A11 P48066 2/20 0.41
SLC6A13 Q9NSD5 2/20 0.41
GABRA1 P14867 1/20 0.41
GABRR1 P24046 1/20 0.41
GABRA4 P48169 1/20 0.41
CCR2 P41597 1/20 0.36
KCNH2 Q12809 1/20 0.36
ACHE P22303 1/20 0.36
HTR6 P50406 1/20 0.36
GBA1 P04062 2/20 0.36
CACNA2D1 P54289 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNB1 Q02641 1/20 0.34
HRH4 Q9H3N8 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3660482 1.00 CHRM5 (0.52) CHRM5ADRA2CSLC6A1GABRA5GABRB2
SCHEMBL14505993 1.00 CHRM5 (0.52) CHRM5ADRA2CSLC6A1GABRA5GABRB2
SCHEMBL29862023 0.98 CHRM5 (0.56) CHRM5ADRA2CSLC6A1GABRA5GABRB2
Hydrochloric Acid SCHEMBL20520976 0.98 CHRM5 (0.50) CHRM5ADRA2CSLC6A1GABRA5GABRB2
Hydrochloric Acid SCHEMBL8449332 0.98 CHRM5 (0.50) CHRM5ADRA2CSLC6A1GABRA5GABRB2
SCHEMBL2462435 0.98 CHRM5 (0.56) CHRM5ADRA2CSLC6A1GABRA5GABRB2
SCHEMBL13950187 0.98 CHRM5 (0.56) CHRM5ADRA2CSLC6A1GABRA5GABRB2
Hydrochloric Acid SCHEMBL20520975 0.98 CHRM5 (0.50) CHRM5ADRA2CSLC6A1GABRA5GABRB2
Hydrochloric Acid SCHEMBL29134438 0.98 CHRM5 (0.50) CHRM5ADRA2CSLC6A1GABRA5GABRB2
SCHEMBL28249891 0.98 CHRM5 (0.56) CHRM5ADRA2CSLC6A1GABRA5GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4045040-A1 NITROGEN CONTAINING BICYCLIC COMPOUNDS Wockhardt Limited (IN) 2022-08-24 EP disclosed
CN-102971291-B Novel amide derivative and use thereof as medicine MITSUBISHI TANABE PHARMA CORP 2015-07-22 CN disclosed
CN-101437819-B Pyridopyrazines and derivatives thereof as alk and c-MET inhibitors CEPHALON INC 2013-06-19 CN disclosed
CN-102971291-A Novel amide derivative and use thereof as medicine MITSUBISHI TANABE PHARMA CORP 2013-03-13 CN disclosed
CN-101456841-B Amide derivative and medicine NIPPON SHINYAKU CO LTD 2012-01-25 CN disclosed
CN-100526298-C Amide derivative and pharmaceutical NIPPON SHINYAKU CO LTD (JP) 2009-08-12 CN disclosed
CN-101456841-A Amide derivative and medicine NIPPON SHINYAKU CO LTD (JP) 2009-06-17 CN disclosed
CN-101437819-A Pyridopyrazines and derivatives thereof as ALK and c-MET inhibitors CEPHALON INC (US) 2009-05-20 CN disclosed
CN-1898208-A Amide derivative and pharmaceutical NIPPON SHINYAKU CO LTD (JP) 2007-01-17 CN disclosed
CN-1041087-C Arylacetamides MERCK PATENT AG (DE) 1998-12-09 CN disclosed