SCHEMBL2745992

SCHEMBL2745992

COc1c(C=Cc2ccc(NS(C)(=O)=O)cc2)cc(-c2c[nH]c(=O)[nH]c2=O)cc1OC(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.55
KIF11 P52732 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
ABL1 P00519 5/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CYP17A1 P05093 1/20 0.33
DPYD Q12882 1/20 0.32
FYN P06241 2/20 0.32
BCR P11274 1/20 0.32
PADI4 Q9UM07 1/20 0.32
TGFBR1 P36897 1/20 0.32
ACVR1 Q04771 1/20 0.32
NFE2L2 Q16236 1/20 0.31
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2745990 1.00 CYP3A4 (0.55) CYP3A4KIF11TRPV1ABL1ALDH1A1
SCHEMBL483525 0.88 CYP3A4 (0.63) CYP3A4KIF11TRPV1ABL1ALDH1A1
SCHEMBL483527 0.88 CYP3A4 (0.63) CYP3A4KIF11TRPV1ABL1ALDH1A1
SCHEMBL2510674 0.85 CYP3A4 (0.54) CYP3A4KIF11TRPV1ABL1ALDH1A1
SCHEMBL2510672 0.85 CYP3A4 (0.54) CYP3A4KIF11TRPV1ABL1ALDH1A1
SCHEMBL482574 0.85 CYP3A4 (0.75) CYP3A4TRPV1ALDH1A1LMNADPYD
SCHEMBL482573 0.85 CYP3A4 (0.75) CYP3A4TRPV1ALDH1A1LMNADPYD
SCHEMBL1764958 0.83 CYP3A4 (0.66) CYP3A4TRPV1ALDH1A1LMNADPYD
SCHEMBL2520555 0.81 CYP3A4 (0.51) CYP3A4ABL1ALDH1A1LMNADPYD
SCHEMBL2520553 0.81 CYP3A4 (0.51) CYP3A4ABL1ALDH1A1LMNADPYD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8178547-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2012-05-15 US disclosed
US-20100158860-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS STEINER SANDRA 2010-06-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100158860-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS RFC1, RRP1B, RRBP1 CYP3A4 978/4885KIF11 4269/4885TRPV1 4760/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.