SCHEMBL27460495

SCHEMBL27460495

O=C1N(OC(=O)C(F)(F)F)c2ccsc2CN1C1CCNCC1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.33
P2RX7 Q99572 1/20 0.31
NOS1 P29475 2/20 0.31
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4782074 0.81 PARP1 (0.42) PARP1
SCHEMBL7831850 0.80 PARP1 (0.35) PARP1
SCHEMBL3964411 0.72 JAK2 (0.36) NOS1NOS2
Trifluoroacetic Acid SCHEMBL3960183 0.70 PARP1 (0.35) PARP1P2RX7
SCHEMBL2212755 0.66 PARP1 (0.45) PARP1
SCHEMBL14141234 0.64 MAPK1 (0.39) PARP1NOS1NOS3NOS2
Trifluoroacetic Acid SCHEMBL3816984 0.59 PARP1 (0.36) PARP1P2RX7
Trifluoroacetic Acid SCHEMBL3085405 0.58 PARP1 (0.52) PARP1
SCHEMBL3279312 0.58 PARP1 (0.49) PARP1
Trifluoroacetic Acid SCHEMBL4782071 0.58 CALCRL (0.48) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1129605-C Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn. THOMAE GMBH DR K (DE) 2003-12-03 CN disclosed
CN-1230196-A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn. THOMAE GMBH DR K (DE) 1999-09-29 CN disclosed