SCHEMBL27460925

SCHEMBL27460925

CCOc1cc2ncc(C#N)c(Nc3cccc(CC)c3)c2cc1OCC

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 15/20 0.77
ERBB2 P04626 13/20 0.77
GAK O14976 2/20 0.61
STK4 Q13043 2/20 0.61
SRC P12931 2/20 0.60
MAP2K1 Q02750 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6383704 0.88 EGFR (0.78) EGFRERBB2STK4SRCMAP2K1
SCHEMBL95052 0.87 EGFR (1.00) EGFRERBB2GAKSTK4
SCHEMBL6382094 0.87 EGFR (0.80) EGFRERBB2GAKSTK4SRC
SCHEMBL6382235 0.87 EGFR (0.80) EGFRERBB2GAKSTK4SRC
SCHEMBL6380499 0.84 EGFR (1.00) EGFRERBB2GAKSRCMAP2K1
SCHEMBL6381507 0.84 EGFR (0.82) EGFRERBB2STK4
SCHEMBL6379850 0.84 EGFR (1.00) EGFRERBB2GAKSRCMAP2K1
SCHEMBL6384856 0.82 EGFR (0.76) EGFRERBB2GAKSRCMAP2K1
SCHEMBL6380110 0.82 EGFR (0.77) EGFRERBB2GAKSRCMAP2K1
SCHEMBL6385549 0.82 EGFR (0.74) EGFRERBB2GAKSRCMAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1121391-C Substituted 3-cyano quinolines AMERICAN CYANAMID CO (US) 2003-09-17 CN claimed
CN-1259125-A Substituted 3-cyanoquinolines AMERICAN CYANAMID CO (US) 2000-07-05 CN claimed