SCHEMBL27468575

SCHEMBL27468575

COc1cc(CC2CNCCN2)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.41
LTA4H P09960 1/20 0.39
PDE4A P27815 2/20 0.38
MAPK1 P28482 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4D Q08499 2/20 0.38
TNF P01375 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
KMT2A Q03164 1/20 0.38
PRMT5 O14744 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL27470245 0.99 HRH3 (0.40) HRH3LTA4HPDE4AMAPK1PDE4B
SCHEMBL2245482 0.89 HRH3 (0.41) HRH3LTA4HPDE4AMAPK1PDE4B
SCHEMBL5270104 0.89 HRH3 (0.41) HRH3LTA4HPDE4AMAPK1PDE4B
Bromide SCHEMBL6132805 0.84 HRH3 (0.41) HRH3LTA4HPDE4AMAPK1PDE4B
SCHEMBL27508444 0.84 HTR2A (0.43) HRH3LTA4HPDE4AMAPK1PDE4B
Hydrochloric Acid SCHEMBL27519893 0.83 HTR2A (0.42) HRH3LTA4HPDE4AMAPK1PDE4B
Bromide SCHEMBL5369378 0.82 HTR2A (0.50) HRH3LTA4H
SCHEMBL27471263 0.82 SSTR1 (0.41) HRH3LTA4H
Bromide SCHEMBL6132803 0.81 HRH3 (0.41) HRH3LTA4HPDE4AMAPK1PDE4B
SCHEMBL28746746 0.79 HRH3 (0.43) HRH3LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1152877-C Piperazine derivatives ����ҩƷ��ҵ��ʽ���� 2004-06-09 CN disclosed
CN-1334812-A Piperazine derivatives FUJISAWA PHARMACEUTICAL CO (JP) 2002-02-06 CN disclosed