SCHEMBL27486209

SCHEMBL27486209

CC(C)C(CCBr)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 1/20 0.46
SLC1A2 P43004 1/20 0.46
SLC1A1 P43005 1/20 0.46
TDP1 Q9NUW8 2/20 0.36
GABRR1 P24046 2/20 0.36
CYP1A2 P05177 1/20 0.36
TP53 P04637 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
SLC7A5 Q01650 1/20 0.35
CHRM1 P11229 1/20 0.33
AKR1A1 P14550 1/20 0.33
CHRM3 P20309 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33
DRD3 P35462 1/20 0.33
SLC6A3 Q01959 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16140111 0.79 SLC1A3 (0.50) SLC1A3SLC1A2SLC1A1TDP1GABRR1
SCHEMBL4610258 0.79
SCHEMBL967949 0.77 CHRM1 (0.52) SLC1A3SLC1A2SLC1A1TDP1TSHR
SCHEMBL1572883 0.77 SLC1A3 (0.48) SLC1A3SLC1A2SLC1A1TDP1GABRR1
SCHEMBL5514417 0.77 SLC1A3 (0.48) SLC1A3SLC1A2SLC1A1TDP1GABRR1
SCHEMBL31544399 0.77 SLC1A3 (0.48) SLC1A3SLC1A2SLC1A1TDP1GABRR1
SCHEMBL31544402 0.77 SLC1A3 (0.48) SLC1A3SLC1A2SLC1A1TDP1GABRR1
SCHEMBL3651519 0.77 CHRM1 (0.52) SLC1A3SLC1A2SLC1A1TDP1TSHR
SCHEMBL21052495 0.77 GABRR1 (0.54) SLC1A3SLC1A2SLC1A1TDP1GABRR1
SCHEMBL188173 0.77 SLC1A3 (0.48) SLC1A3SLC1A2SLC1A1TDP1GABRR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1183107-C Alkynyl containing hydroxamic acid compounds as TACE inhibitors ���Ͽع����޹�˾ 2005-01-05 CN disclosed
CN-1337945-A Alkynyl containing hydroxamic acid compounds as TACE inhibitors AMERICAN CYANAMID CO (US) 2002-02-27 CN disclosed
CN-1283183-A Hydroxamic and carboxylic acid derivatives having MMP and TNF inhibitory activity DARWIN DISCOVERY LTD (GB) 2001-02-07 CN disclosed
CN-1227540-A Hydroxamic and carboxylic acid derivatives having MMP and TNF inhibitory activity DARWIN DISCOVERY CO LTD (GB) 1999-09-01 CN disclosed