SCHEMBL27488281

SCHEMBL27488281

CCCCCNS(=O)(=O)c1cccc2ccccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.72
CYP3A4 P08684 5/20 0.72
CYP2C19 P33261 5/20 0.72
CYP2C9 P11712 4/20 0.72
ALDH1A1 P00352 3/20 0.72
SCN1A P35498 2/20 0.72
SCN2A Q99250 2/20 0.72
SCN3A Q9NY46 2/20 0.72
KDM4E B2RXH2 2/20 0.72
HSD17B10 Q99714 1/20 0.72
TP53 P04637 3/20 0.68
TDP1 Q9NUW8 3/20 0.68
MEN1 O00255 2/20 0.68
TSHR P16473 2/20 0.68
KMT2A Q03164 2/20 0.68
RECQL P46063 1/20 0.62
NPY5R Q15761 5/20 0.60
CA12 O43570 2/20 0.59
CA9 Q16790 2/20 0.59
HTR7 P34969 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29141930 0.98 CYP3A4 (0.74) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL3698543 0.95 CYP3A4 (0.69) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL3680789 0.89 CYP3A4 (0.64) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
Bromide SCHEMBL28238291 0.86 CYP3A4 (0.61) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL23072066 0.85 CYP3A4 (0.68) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL8024067 0.85 CYP3A4 (0.97) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL29941333 0.84 SCN1A (0.56) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL28062482 0.84 CYP3A4 (0.62) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL30306219 0.84 CYP3A4 (1.00) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL6753337 0.84 CYP3A4 (1.00) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101151249-B Cyclopentapyridine and tetrahydroquinoline derivatives PFIZER PRODUCTS INC. (US) 2011-04-06 CN disclosed
CN-101151249-A Cyclopentapyridine and tetrahydroquinoline derivatives PFIZER (US) 2008-03-26 CN disclosed
CN-1745074-A 5-HT receptor ligands and uses thereof PFIZER PROD INC (US) 2006-03-08 CN disclosed
CN-1212315-C Coffee acyl naphthalene sulfonamides compound and method for preparing the same and anti HIV conformity enzyme action UNIV SHANDONG (CN) 2005-07-27 CN disclosed
CN-1212315-C Coffee acyl naphthalene sulfonamides compound and method for preparing the same and anti HIV conformity enzyme action UNIV SHANDONG (CN) 2005-07-27 CN disclosed
CN-1630645-A 5-HT receptor ligands and uses thereof PFIZER (US) 2005-06-22 CN disclosed
CN-1482116-A Coffee acyl naphthalene sulfonamides compound and method for preparing the same and anti HIV conformity enzyme action 山东大学 2004-03-17 CN disclosed