SCHEMBL27508331

SCHEMBL27508331

COCCC1[CH]CCNC1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL293097 0.78
SCHEMBL27644423 0.73 KCNA3 (0.41) SLC6A2SLC6A4SLC6A3
SCHEMBL27482999 0.73
SCHEMBL27467944 0.70
SCHEMBL16288185 0.69
SCHEMBL2430952 0.69 POLB (0.31)
SCHEMBL2917543 0.69 CYP2D6 (0.31) CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL4539262 0.69
SCHEMBL27515837 0.67
SCHEMBL10103535 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1322202-A Quinazoline derivatives ASTRA ZENECA N V (SE) 2001-11-14 CN claimed
CN-100360505-C Quinazoline derivatives as angiogenesis inhibitors ASTRAZENECA AB (SE) 2008-01-09 CN disclosed
CN-1315822-C Quinoline derivatives having VEGF inhibiting activity STRAZENECA AB (SE) 2007-05-16 CN disclosed
CN-1252065-C Cinnoline compounds ASTRAZENECA AB (SE) 2006-04-19 CN disclosed
CN-1245402-C indole derivatives, process for their preparation, pharmaceutical compositions containing them and their use ASTRAZENECA AB (SE) 2006-03-15 CN disclosed
CN-1597667-A Quinazoline derivatives as angiogenesis inhibitors ASTRAZENECA AB (SE) 2005-03-23 CN disclosed
CN-1167422-C Quinazoline derivatives as angiogenesis inhibitors 2004-09-22 CN disclosed
CN-1161352-C Quinazoline derivatives 2004-08-11 CN disclosed
CN-1468230-A Compound (I) 2004-01-14 CN disclosed
CN-1446212-A Quinoline derivatives having VEGF inhibiting activity STRAZENECA AB (SE) 2003-10-01 CN disclosed
CN-1446214-A Cinnoline compounds ASTRAZENECA AB (SE) 2003-10-01 CN disclosed
CN-1346271-A Quinazoline derivatives as angiogenesis inhibitors ASTRAZENECA UK LTD (SE) 2002-04-24 CN disclosed
CN-1322202-A Quinazoline derivatives ASTRA ZENECA N V (SE) 2001-11-14 CN disclosed