SCHEMBL27509869

SCHEMBL27509869

O=C(NCc1ccc(CN(C2CCNCC2)C2CCCc3cccnc32)cc1)c1ccncc1Cl

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 19/20 0.42
CYP3A4 P08684 8/20 0.42
CYP2D6 P10635 8/20 0.42
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27509522 0.94 CXCR4 (0.39) CXCR4CYP3A4CYP2D6
SCHEMBL4063134 0.91 CXCR4 (0.41) CXCR4CYP3A4CYP2D6HDAC1HDAC6
SCHEMBL4069138 0.87 CXCR4 (0.40) CXCR4CYP3A4CYP2D6HDAC1HDAC6
SCHEMBL4062979 0.85 CXCR4 (0.40) CXCR4CYP3A4CYP2D6
SCHEMBL27509870 0.84 HDAC1 (0.42) CXCR4CYP3A4CYP2D6HDAC1HDAC6
SCHEMBL4066923 0.83 CXCR4 (0.41) CXCR4CYP3A4CYP2D6HDAC1HDAC6
SCHEMBL27529288 0.82 CXCR4 (0.47) CXCR4CYP3A4CYP2D6
SCHEMBL4061365 0.82 HDAC1 (0.40) CXCR4CYP3A4CYP2D6HDAC1HDAC6
SCHEMBL4072213 0.80 CXCR4 (0.39) CXCR4CYP3A4CYP2D6
SCHEMBL27533357 0.80 CXCR4 (0.45) CXCR4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1237061-C Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2006-01-18 CN disclosed
CN-1458929-A Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2003-11-26 CN disclosed