SCHEMBL27529338

SCHEMBL27529338

CC1=CN=C(CN(Cc2ccc(CNC(=O)c3ccnc(Cl)c3)cc2)C2CCCc3cccnc32)C1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 17/20 0.42
CYP2D6 P10635 9/20 0.42
CYP3A4 P08684 8/20 0.42
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27509541 0.94 CXCR4 (0.42) CXCR4CYP2D6CYP3A4
SCHEMBL27509527 0.88 CXCR4 (0.40) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27510609 0.87 CXCR4 (0.41) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL4062767 0.86 CXCR4 (0.44) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27511684 0.85 CXCR4 (0.41) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27529336 0.85 CXCR4 (0.45) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27578502 0.85 CXCR4 (0.41) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27529290 0.84 CXCR4 (0.47) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27578506 0.84 CXCR4 (0.42) CXCR4CYP2D6CYP3A4HDAC1HDAC6
SCHEMBL27529298 0.84 CXCR4 (0.41) CXCR4CYP2D6CYP3A4HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1237061-C Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2006-01-18 CN disclosed
CN-1458929-A Chemokine receptor binding heterocyclic compounds ANORMED INC (CA) 2003-11-26 CN disclosed