SCHEMBL27537751

SCHEMBL27537751

Cc1cc(C(=O)O)c(NC(=O)OC(C)(C)C)c(C(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LCK P06239 7/20 0.44
KDM4E B2RXH2 1/20 0.43
ATR Q13535 1/20 0.43
METAP2 P50579 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
CSNK2A1 P68400 1/20 0.37
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108498 0.92 LCK (0.50) LCKKDM4EATRMETAP2CA12
SCHEMBL27969586 0.90 LCK (0.44) LCKKDM4EATRMETAP2MEN1
SCHEMBL8651106 0.81 ATR (0.47) LCKKDM4EATRCA12CA1
SCHEMBL3131919 0.81 LCK (0.60) LCKCA12CA1CA9NFKB1
SCHEMBL27852761 0.81 MEN1 (0.56) METAP2CA12CA1CSNK2A1MEN1
SCHEMBL19678555 0.78 ATR (0.39) LCKATRCA12CA1CA9
SCHEMBL108868 0.78 ATR (0.51) LCKKDM4EATRCA12CA1
SCHEMBL12884719 0.76 POLB (0.53) LCKKDM4EATRMEN1KMT2A
SCHEMBL4289283 0.76 LCK (0.40) LCKATRCA12CA1CA9
SCHEMBL12731272 0.76 ATR (0.49) LCKKDM4EATRGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101074242-A Cells accumulation for sphosphonate analogs of HIV protease inhibitor compound and the same compound GILEAD SCIENCES INC (US) 2007-11-21 CN disclosed
CN-1313472-C Cellular Accumulation of Phosphonate Analogs of HIV Protease Inhibitor Compounds and Such Compounds GILEAD SCIENCES INC (US) 2007-05-02 CN disclosed
CN-1649885-A Cellular Accumulation of Phosphonate Analogs of HIV Protease Inhibitor Compounds and Such Compounds GILEAD SCIENCES INC (US) 2005-08-03 CN disclosed