SCHEMBL27540539

SCHEMBL27540539

Cc1[nH]nc(-c2cccc(Br)c2)c1-c1ccncc1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.57
LRRK2 Q5S007 17/20 0.56
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
CNR1 P21554 1/20 0.45
CNR2 P34972 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27741317 0.84 IKBKB (0.66) IKBKBLRRK2CNR1CNR2GPR55
SCHEMBL5450217 0.83 LRRK2 (0.56) LRRK2MAPK11MAPK14
SCHEMBL2479766 0.83 MAPK14 (0.44) IKBKBLRRK2MAPK11MAPK14
SCHEMBL7852194 0.83 MAPK11 (0.59) LRRK2MAPK11MAPK14
SCHEMBL5446476 0.82 IKBKB (0.57) IKBKBLRRK2CNR1CNR2GPR55
SCHEMBL14519374 0.82 LRRK2 (0.60) LRRK2
SCHEMBL5255653 0.81 LRRK2 (0.54) LRRK2MAPK11MAPK14
SCHEMBL14521814 0.80 MAPK14 (0.42) IKBKBLRRK2MAPK11MAPK14
SCHEMBL5449961 0.78 LRRK2 (0.54) LRRK2MAPK14
SCHEMBL14519600 0.77 MAPK14 (0.52) MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1264377-A Substituted pyrazoles as P38 kinase inhabitors SEARLE & CO (US) 2000-08-23 CN claimed
CN-1273603-A Attenuated respiratory syncytial virus AMERICAN CYANAMID CO (US) 2000-11-15 CN disclosed