SCHEMBL27584530

SCHEMBL27584530

C#CCCCn1c(Cc2cc(OC)c(OC)c(OC)c2Cl)nc2c(C(N)=O)nc(F)nc21

nearest known ligand 0.77

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 18/20 0.77
HSP90AB1 P08238 18/20 0.77
ERBB2 P04626 6/20 0.61
HSP90B1 P14625 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27584533 0.88 HSP90AA1 (0.76) HSP90AA1HSP90AB1ERBB2
SCHEMBL2604977 0.87 HSP90AA1 (1.00) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL10149974 0.81 HSP90AA1 (0.87) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL4462613 0.78 HSP90AA1 (0.77) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL30583139 0.78 HSP90AA1 (0.77) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL27602471 0.77 HSP90AA1 (0.59) HSP90AA1HSP90AB1ERBB2
SCHEMBL23819778 0.77 HSP90AA1 (0.81) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL27602461 0.76 HSP90AA1 (0.60) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL1864541 0.76 HSP90AA1 (1.00) HSP90AA1HSP90AB1ERBB2HSP90B1
SCHEMBL23450478 0.76 HSP90AA1 (0.79) HSP90AA1HSP90AB1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101928288-A Small molecule compositions for binding to HSP90 SLOAN KETTERING INST CANCER 2010-12-29 CN disclosed
CN-1501928-A Small molecule compositions that bind HSP90 斯隆-凯特林癌症研究所 2004-06-02 CN disclosed