SCHEMBL27591978

SCHEMBL27591978

COc1ccc(-c2nc(N)nc([S+](C)[O-])c2C#N)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 15/20 0.42
ADORA2A P29274 13/20 0.39
ADORA2B P29275 5/20 0.38
MAPT P10636 4/20 0.34
RXFP1 Q9HBX9 1/20 0.34
KDM4E B2RXH2 3/20 0.32
ALDH1A1 P00352 3/20 0.32
MAPK1 P28482 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
GAA P10253 2/20 0.31
PKM P14618 2/20 0.31
HPGD P15428 2/20 0.31
LMNA P02545 1/20 0.31
GLA P06280 1/20 0.31
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ALOX12 P18054 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6440596 0.88 KDM4E (0.42) ADORA1ADORA2AADORA2BMAPTKDM4E
SCHEMBL6442849 0.85 ADORA1 (0.37) ADORA1ADORA2AADORA2BMAPTRXFP1
SCHEMBL6440737 0.84 ADORA1 (0.36) ADORA1ADORA2AADORA2BMAPTKDM4E
SCHEMBL6444418 0.82 ADORA1 (0.36) ADORA1ADORA2AADORA2BMAPTKDM4E
SCHEMBL6444885 0.78 ADORA2A (0.61) ADORA1ADORA2AADORA2BMAPTKDM4E
SCHEMBL6442282 0.78 MAPT (0.57) ADORA1ADORA2AADORA2BMAPTRXFP1
SCHEMBL6441010 0.76 GRM4 (0.40) ADORA1ADORA2AADORA2BMAPTKDM4E
SCHEMBL6440809 0.76 ADORA2A (0.66) ADORA1ADORA2AADORA2BMAPTKDM4E
SCHEMBL6442913 0.74 ADORA1 (0.36) ADORA1ADORA2AADORA2BKDM4E
SCHEMBL6441176 0.74 ADORA1 (0.36) ADORA1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1438890-A Adenosine receptor modulators HOFFMANNLA ROCHE AG F (CH) 2003-08-27 CN disclosed