SCHEMBL27592220

SCHEMBL27592220

COC(=O)c1ccccc1NS(=O)(=O)C1CCCC=C1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
KDM4E B2RXH2 8/20 0.46
ALDH1A1 P00352 5/20 0.46
TLR4 O00206 4/20 0.46
HSD17B10 Q99714 3/20 0.45
HPGD P15428 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
RECQL P46063 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.43
KDM1A O60341 1/20 0.43
MRGPRX1 Q96LB2 1/20 0.43
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
POLB P06746 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27576686 0.89 TLR4 (0.57) TSHRKDM4EALDH1A1TLR4HSD17B10
SCHEMBL871405 0.87 TLR4 (0.62) TSHRKDM4EALDH1A1TLR4HSD17B10
SCHEMBL872228 0.82 TLR4 (0.64) TSHRKDM4EALDH1A1TLR4HSD17B10
SCHEMBL27592263 0.81 TLR4 (0.48) TSHRKDM4EALDH1A1TLR4KMT2A
SCHEMBL6053601 0.81 TLR4 (0.52) TSHRKDM4ETLR4SMN1; SMN2MRGPRX1
SCHEMBL27573690 0.81 TLR4 (0.52) TSHRALDH1A1TLR4MEN1GAA
SCHEMBL27573738 0.80 HPGD (0.47) TSHRALDH1A1TLR4HPGDMEN1
SCHEMBL27883083 0.79 TLR4 (0.41) KDM4EALDH1A1TLR4HPGDSMN1; SMN2
SCHEMBL27592264 0.78 TLR4 (0.60) TSHRKDM4EALDH1A1TLR4HSD17B10
SCHEMBL28159696 0.77 TLR4 (0.48) TSHRALDH1A1TLR4NPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102821763-B Compound for inhibiting peripheral nerve disorder induced by anticancer agent 武田药品工业株式会社 2017-09-22 CN disclosed
CN-101212986-B Stable emulsified composition TAKEDA PHARMACEUTICAL 2015-01-14 CN disclosed
CN-102821763-A Compound for inhibiting peripheral nerve disorder induced by anticancer agent TAKEDA PHARMACEUTICAL 2012-12-12 CN disclosed
CN-102670503-A Stable emulsion composition TAKEDA PHARMACEUTICAL 2012-09-19 CN disclosed
CN-1416341-B Stable emulsion compositions TAKEDA CHEMICAL INDUSTRIES LTD 2010-05-05 CN disclosed
CN-101212986-A stable emulsified composition TAKEDA PHARMACEUTICAL (JP) 2008-07-02 CN disclosed
CN-1416341-A Stable emulsion compsns TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-07 CN disclosed