SCHEMBL27596754

SCHEMBL27596754

Nc1nc(N(S)C=O)c2ncn(Cc3ccccc3F)c2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.55
ADORA1 P30542 4/20 0.55
PDE4A P27815 5/20 0.45
PDE4B Q07343 5/20 0.45
PDE4C Q08493 5/20 0.45
PDE4D Q08499 5/20 0.45
PDE5A O76074 3/20 0.44
PDE1A P54750 3/20 0.44
PDE1B Q01064 3/20 0.44
PDE1C Q14123 3/20 0.44
HDAC6 Q9UBN7 2/20 0.43
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738116 0.83 ADORA2A (0.60) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL3269795 0.79 ADORA2A (0.64) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL9738574 0.79 ADORA2A (0.66) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL11014088 0.76 PDE4A (0.61) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL3269162 0.74 ADORA2A (0.60) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL3268278 0.74 ADORA2A (0.60) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL9739023 0.74 PDE4A (0.72) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL3268280 0.74 ADORA2A (0.57) ADORA2AADORA1PDE4APDE4BPDE4C
SCHEMBL3269399 0.71 ADORA2A (1.00) ADORA2AADORA1ADORA3ADORA2B
SCHEMBL3272538 0.71 ADORA2A (0.56) ADORA2AADORA1PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1617871-A Purine derivatives as purinergic receptor antagonists VERNALIS RES LTD (GB) 2005-05-18 CN disclosed