SCHEMBL27612367

SCHEMBL27612367

CC(C)Oc1ccc(Nc2nc(Cl)ncc2F)cc1Cl.CNC(=O)c1cccc(NOC)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.50
SYK P43405 7/20 0.49
BCL6 P41182 4/20 0.46
BTK Q06187 1/20 0.45
NCOR2 Q9Y618 1/20 0.44
EGFR P00533 4/20 0.44
PTK2 Q05397 1/20 0.44
KCNQ3 O43525 1/20 0.42
KCNQ2 O43526 1/20 0.42
ERBB2 P04626 1/20 0.42
ITK Q08881 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27612425 0.88 EGFR (0.53) SCN9ASYKBTKEGFRKCNQ3
SCHEMBL2302190 0.83 SCN9A (0.58) SCN9ASYK
SCHEMBL2103835 0.82 BCL6 (0.60) SYKBCL6NCOR2EGFRITK
SCHEMBL27612600 0.76 SYK (0.66) SYKBCL6EGFRITK
SCHEMBL12519774 0.75 MAPK1 (0.54) SYKEGFRITK
SCHEMBL2061066 0.75 ALK (0.55) SCN9A
SCHEMBL657489 0.74 POLB (0.53) SYKBCL6NCOR2EGFRPTK2
SCHEMBL658038 0.73 BCL6 (0.71) SYKBCL6NCOR2EGFRERBB2
SCHEMBL267189 0.72 EGFR (0.50) SCN9ASYKBTKEGFR
SCHEMBL27631540 0.71 SYK (0.54) SYKBCL6NCOR2EGFRPTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1678321-A Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds RIGEL PHARMACEUTICALS INC (US) 2005-10-05 CN disclosed